I-Amino Tadalafil powder umenzi we-CAS No.: 385769-84-6 98% ubumsulwa min.zokongeza izithako
IiParameters zeMveliso
| Igama lemveliso | Amino Tadalafil |
| Elinye igama | (6R,12aR)-2-Amino-6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[ 3,4-b]indole-1,4-dione;AminoTadalafil(6R,12Ar)-2-Amino-6-(1,3-Benzodioxol-5-Yl)-2,3,6,7,12,12A -Hexahydropyrazino [1',2':1,6]Pyrido[3,4-B]Indole-1,4-Dione;(6R,12aR) -2-Amino-6-(benzo[d][1,3] ]dioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indol-1,4-dione;(6R ,12aR) -2-amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,12,12a-tetrahydropyrazino[1',2':1,6]pyrido[3] ,4-b]indole-1,4(6H,7H)-dione |
| Inombolo yeCAS. | 385769-84-6 |
| Ifomula yemolekyuli | I-C21H18N4O4 |
| Ubunzima bemolekyuli | 390.39 |
| Ubunyulu | 98.0% |
| Imbonakalo | Umgubo omhlophe ukuya kumhlophe |
| Isicelo | I-Dietary Supplement Raw Material |
Intshayelelo yemveliso
I-Amino Tadalafil i-compound efana ne-Tadalafil, kunye namanye amaqela asebenzayo kwisakhiwo sayo athatyathwa ngamaqela e-amino.I-PDE5 inhibitor kwaye ineempembelelo ze-pharmacological ezifana neTadalafil.Isetyenziswa ikakhulu kunyango lwe-male erectile dysfunction (ED).Xa kuthelekiswa neTadalafil, i-Amino Tadalafil inesantya esincinci se-metabolism emzimbeni, kwaye ngoko ke ingaba nefuthe elihlala ixesha elide.
Uphawu
(1) Ukukhetha okuphezulu: I-Amino Tadalafil inokukhethwa okuphezulu kwe-PDE5, kunye nobudlelwane obuphezulu kakhulu be-PDE5 kunezinye i-PDE subtypes.Oku kuthetha ukuba i-Amino Tadalafil inokuthintela ngokufanelekileyo umsebenzi we-PDE5 enzyme, ukukhuthaza ukuhamba kwegazi kwizitho zokuzala zesilisa kunye nokuphucula iimpawu ze-erectile dysfunction (ED).
(2) Impembelelo ehlala ixesha elide: I-Amino Tadalafil inesantya esincinci se-metabolism emzimbeni, esivumela ukuba sivelise umphumo we-pharmacological wexesha elide, elihlala kwiiyure ze-36.Oku kwenza i-Amino Tadalafil isilwanyana sonyango se-ED eside, esingafuneki ukuba sithathwe rhoqo.
(3) Imiphumo emibi embalwa: I-Amino Tadalafil ineempembelelo ezincinci xa kuthelekiswa neTadalafil, njengentloko, kunye nokuphazamiseka kwesisu.Ngenxa yokukhethwa kwayo okuphezulu, i-Amino Tadalafil inokuphepha ngokufanelekileyo ukusebenzisana nezinye ii-PDE subtypes, ukunciphisa iziganeko zemiphumo emibi.
(4) Amathuba okusetyenziswa ngokubanzi: Ngaphandle kokunyanga i-ED, i-Amino Tadalafil ingasetyenziselwa ukuphatha ezinye izifo ezifana ne-pulmonary arterial hypertension.Oku kwenza i-Amino Tadalafil ibe nethemba elibanzi lesicelo kwixesha elizayo.
Usetyenziso
I-Amino Tadalafil yi-compound ephuhliswe kwiminyaka yamuva, enesakhiwo esifana neTadalafil, kodwa amanye amaqela kwisakhiwo sayo athatyathwa ngamaqela e-amino.Okwangoku, i-Amino Tadalafil ayivunywanga ukusetyenziswa kwezonyango, ngoko ke isicelo sayo kwinkalo yezonyango silinganiselwe.Nangona kunjalo, ezinye izifundo zibonise ukuba le khompawundi inamandla amakhulu okusetyenziswa.
I-Amino Tadalafil yi-PDE5 inhibitor, enefuthe elifanayo le-pharmacological njengeTadalafil.Inokuphucula iimpawu ze-erectile dysfunction (ED) ngokukhuthaza ukuhamba kwegazi kwizitho zokuzala zesilisa ngokuthintela umsebenzi we-PDE5 enzyme.Xa kuthelekiswa neTadalafil, i-Amino Tadalafil inesantya esincinci semetabolism emzimbeni, enokuthi ibe nefuthe elihlala njalo.Oku kwenza i-Amino Tadalafil ibe namandla amakhulu kunyango lwe-ED.
Ukongeza, i-Amino Tadalafil inokusetyenziselwa ukunyanga ezinye izifo, ezinje nge-pulmonary arterial hypertension.Olunye uphando lubonise ukuba i-PDE5 inhibitors inokwandisa imithwalo yegazi ye-pulmonary, ngaloo ndlela iphucula iimpawu zezigulane ezine-pulmonary arterial hypertension.Ngenxa yokuba i-Amino Tadalafil inefuthe elifanayo le-pharmacological njenge-Tadalafil, ingasetyenziselwa ukunyanga uxinzelelo lwegazi lwe-pulmonary.
Ngokubanzi, i-Amino Tadalafil inamandla okwenza isicelo, kodwa izilingo ezininzi zeklinikhi ziyafuneka ukuze kuqinisekiswe ukhuseleko kunye nokusebenza kakuhle.Ukuba ezi zilingo zivelisa iziphumo ezilungileyo, i-Amino Tadalafil inokuba liyeza elitsha kunyango lwe-ED kunye ne-pulmonary arterial hypertension, ebonelela ngeendlela ezininzi zonyango koogqirha bezonyango kunye nezigulane.
