ibhena_yephepha

imveliso

Umenzi womgubo weFasoracetam Inombolo yeCAS: 110958-19-5 Ubumsulwa obuyi-99% ubuncinane bezithako ezongezelelweyo

Inkcazo emfutshane:

Ikhemikhali iFasoracetam sisiyobisi esenziweyo esikwiklasi yamachiza ebizwa ngokuba yi-dihydropyridine pyrrolidone class.


Iinkcukacha zeMveliso

Iithegi zeMveliso

Ividiyo yeMveliso

Iiparamitha zeMveliso

Igama lemveliso

I-Fasoracetam

Elinye igama

I-FASORACETAM;

(5R)-5-(piperidine-1-carbonyl)-2-pyrrolidone;

(5R)-5-(piperidine-1-carbonyl)pyrrolidin-2-nye;

(5R)-5-piperidin-1-ylcarbonylpyrrolidin-2-nye

Inombolo ye-CAS

110958-19-5

Ifomula yemolekyuli

C10H16N2O2

Ubunzima be-molecular

196.25

Ubunyulu

99.0%

Inkangeleko

Umgubo omhlophe wekristale

Ukupakisha

1 kg/ibhegi 25kg/igubu

Isicelo

I-Nootropic

Intshayelelo yemveliso

I-Fasoracetam, yikhompawundi ye-nootropic eyaqalwa ukuphuhliswa eJapan. Ifana ngendlela efanayo nezinye iintlobo ze-racemates ezifana ne-piracetam, kodwa ibonisa iimpawu zesenzo ezizodwa. I-Fasoracetam kucingelwa ukuba ilawula iziphumo zee-neurotransmitters ezahlukeneyo engqondweni, kubandakanya iinkqubo ze-GABA, i-glutamatergic, kunye ne-cholinergic. Ngokuchaphazela ukukhululwa kunye nokufunxwa kwezi neurotransmitters, i-fasoracetam inokuphucula imisebenzi yengqondo efana nokuqwalaselwa, ukuhlanganiswa kwememori, kunye nokucubungula ulwazi. Uphando kunye nobungqina be-anecdotal bubonisa ukuba i-fasoracetam inokubonelela ngeenzuzo ezininzi zengqondo. Enye yeziphumo zayo eziphambili kukuphucula ukugxila kunye nexesha lokugxila, okwenza ukuba ibe luncedo kwabo banengxaki yokuphazamiseka kwengqondo okanye ukuphazamiseka kwengqondo (ADD/ADHD). Izifundo zokuqala zibonise iziphumo ezithembisayo, ezibonisa amandla e-fasoracetam okuphucula ingqalelo, ukunciphisa ukunyanzeliswa kunye nokuphucula ulawulo lwengqondo. Ukongeza, izifundo zezilwanyana zibonisa ukuba i-Fasoracetam iphucula amandla exesha elide, inkqubo enxulumene nokwakheka kwememori kunye ne-synaptic plasticity.

Uphawu

(1) Ubunyulu obuphezulu: I-Fasoracetam inokufumana iimveliso ezinyulu obuphezulu ngokusebenzisa iinkqubo zokuvelisa ezicociweyo. Ubunyulu obuphezulu buthetha ukufumaneka ngcono kwezinto eziphilayo kunye neempendulo ezimbalwa ezimbi.

(2) Ukhuseleko: Izifundo zibonise ukuba i-fasoracetam idla ngokunyamezelwa kakuhle kwaye ayibonisi miphumo mibi xa isetyenziswa ngaphakathi kweedosi ezicetyiswayo.

(3) Uzinzo: I-Fasoracetam izinzile kakuhle kwaye inokugcina umsebenzi wayo kunye nesiphumo phantsi kweemeko ezahlukeneyo kunye neemeko zokugcina.

Izicelo

I-Fasoracetam ivele njengesixhobo esinomdla esinamandla okuphucula izakhono zokuqonda, ngakumbi inkumbulo, ingqalelo, kunye nokufunda, kwaye ingasetyenziswa njengesongezelelo sokutya. Le mveliso isebenza njengesiphuculi senkumbulo ngokuvuselela ii-receptors ze-glutamate ze-metabolic. Kwintsimi yebhayoloji, i-Fasoracetam ikwasetyenziswa njengesithinteli esikhethiweyo sokufunda iinkqubo zebhayoloji ezifana nokubonisa iiseli kunye ne-apoptosis.


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