iphepha_ibhena

imveliso

Coluracetam powder umenzi CAS No.: 135463-81-9 99% ubunyulu min.zokongeza izithako

Inkcazelo emfutshane:

I-Coluracetam ilungu lentsapho ye-racetam ye-nootropic compounds kwaye yaziwa nangokuthi yi-MKC-231.Yaphuhliswa yiKobe Pharmaceutical Company eJapan ngenjongo yokunyanga iAD kunye nokuphazamiseka kwengqondo.


Iinkcukacha zeMveliso

Iithegi zeMveliso

IiParameters zeMveliso

Igama lemveliso

I-Coluracetam

Elinye igama

MKC-231;

I-2-oxo-N-(5,6,7,8-tetrahydro-2,3-dimethyl-furo[2,3-b]quinolin-4-yl)-1-pyrrolidineacetamide

Inombolo yeCAS.

135463-81-9

Ifomula yemolekyuli

I-C19H23N3O3

Ubunzima bemolekyuli

341.4

Ubunyulu

99.0%

Imbonakalo

Umgubo omhlophe

Isicelo

I-Dietary Supplement Raw Material

Intshayelelo yemveliso

I-Coluracetam ilungu lentsapho ye-racetam ye-nootropic compounds kwaye yaziwa nangokuthi yi-MKC-231.Yaphuhliswa yiKobe Pharmaceutical Company eJapan ngenjongo yokunyanga iAD kunye nokuphazamiseka kwengqondo.

Indlela echanekileyo yesenzo se-Coluracetam ayiqondwa ngokupheleleyo, kodwa kukholelwa ukuba ngokuyinhloko isebenza ngokumodareyitha inkqubo ye-cholinergic.Kucingelwa ukuba ukwandisa amanqanaba e-acetylcholine, i-neurotransmitter engundoqo kwingqondo ehambelana ngokusondeleyo nokufunda kunye nemisebenzi yememori.I-Coluracetam inokufezekisa oku ngokunyusa inani kunye nomsebenzi we-choline uptake transporters, ekhokelela ekuphuculweni kokukhululwa kwe-acetylcholine kunye nokuhanjiswa kwesignali ephuculweyo phakathi kwe-neurons.

Nangona uphando nge-Coluracetam lusanqongophele, ezinye iimvavanyo zangaphambili kunye nezifundo zezilwanyana ziye zaphakamisa iziphumo ezinokuthi zibe ne-neuroprotective kunye ne-cognitive-pregnitive.Olunye uphando lufumene ukuba i-Coluracetam inophuculo oluthile lokukhubazeka kwememori kwiimodeli ze-AD.

Ngokumalunga nophando lweklinikhi, izifundo kwi-Coluracetam zijolise kakhulu kwiimvavanyo zezilwanyana kunye nezilingo zabantu bokuqala.Uphando olongezelelekileyo kunye nobungqina bufunekayo ukuze kuqinisekiswe ukhuseleko kunye nokusebenza kwalo ebantwini.Okwangoku, i-Coluracetam ayivunywanga ukusetyenziswa kweklinikhi, kodwa isetyenziswa ngokubanzi njengesongezelelo se-nootropic sokuphucula ingqiqo kwamanye amazwe.

Ngokuphathelele ukhuseleko, kukho idatha elinganiselweyo yophando ekhoyo kwimiphumo emibi kunye nobungozi bexesha elide le-Coluracetam.Ngokusekelwe kulwazi lwangoku, i-Coluracetam ngokuqhelekileyo ithathwa njengekhuselekile, kodwa isacetyiswa ukuba udibane nochwepheshe bezempilo, ngakumbi ukuba unayo nayiphi na imeko yezempilo okanye uthatha amanye amayeza, ngaphambi kokuba uyisebenzise.

Isishwankathelo, i-Coluracetam yi-compound ye-nootropic efundwayo ngenxa yokukwazi kwayo ukunyanga i-AD kunye nokuphazamiseka kwengqondo.Ngelixa uphando oluthile lwakwangoko lucebisa ukuphuculwa kwengqondo kunye neziphumo ze-neuroprotective, izifundo ezingaphezulu ziyafuneka ukuseka ukusebenza kokwenyani kunye nokhuseleko.

Uphawu

(1) Ukuhlanjululwa okuphezulu: I-Coluracetam ilungiselelwe ngokusebenzisa ukukhutshwa okuphezulu kunye neenkqubo zokuvelisa, ukuqinisekisa umgangatho ophezulu wokucoceka.Oku kucoceka kuphezulu kunegalelo ekuphuculweni kwe-bioavailability kunye nokunciphisa ukwenzeka kokusabela okubi.

(2) Ukhuseleko: I-Coluracetam ithathwa njengekhuselekile ukuba isetyenziswe ngabantu.Uphononongo olubanzi lubonakalise ubutyhefu bayo obuphantsi kunye neziphumo ebezingalindelekanga ezincinci kuluhlu lwedosi ecetyiswayo.

(3) Ukuzinza: Amalungiselelo e-Coluracetam abonisa ukuzinza okuhle kakhulu, ukugcina umsebenzi wabo kunye nokusebenza phantsi kweemeko ezahlukeneyo zokusingqongileyo kunye nokugcinwa.Oku kuzinza kuqinisekisa ukusebenza okungaguqukiyo kunye nokuthembekileyo ekuhambeni kwexesha.

(4) Ukukhutshwa ngokukhawuleza: I-Coluracetam ithathwa ngokukhawuleza ngumzimba womntu.Ekungeneni, ngokukhawuleza ingena egazini ngokusebenzisa i-intestinal tract kwaye isasaze ngokufanelekileyo kwii-tissue ezahlukeneyo kunye namalungu, iququzelele imiphumo efunwayo.

(5) Ukuphuculwa kwengqondo: I-Coluracetam iyaziwa ngokukwazi ukuphucula umsebenzi wokuqonda, kubandakanywa nokuphuculwa kwememori, amandla okufunda kunye nokugxila.Ihlala ifunwa ngabantu abajonge ukukhulisa ukusebenza kwabo kwengqondo.

(6) Iimpembelelo ze-Neuroprotective: Uphando lubonisa ukuba i-Coluracetam ingaba neepropati ze-neuroprotective, ezinokukunceda ukukhusela ekunciphiseni kwengqondo enxulumene neminyaka kunye nokuxhasa impilo yonke yengqondo.

(7) Unyango olunokubakho kwi-Cognitive Disorders: I-Coluracetam ibonisa isithembiso njengendlela yonyango enokubakho kwiingxaki zengqondo, ezifana nesifo se-Alzheimer kunye nezinye iimeko ze-neurodeergenerative.Nangona kunjalo, uphando olongezelelweyo luyafuneka ukuze kuqondwe ngokupheleleyo ukusebenza kwalo ekunyangeni ezi meko zikhethekileyo.

Usetyenziso

I-Coluracetam okwangoku isetyenziswa kwizicelo ezahlukeneyo kwaye ibonisa amathemba athembisayo kwixesha elizayo.Isetyenziswa ikakhulu njengesongezo sokuphucula ingqondo, efunwa ngabantu abafuna ukuphucula inkumbulo yabo, ukugxila, kunye nobuchule bokufunda.Ukukwazi kwekhompawundi ukulungelelanisa inkqubo ye-cholinergic kukholelwa ukuba negalelo kwimiphumo yokuphucula ingqondo.

Ukongeza kwizicelo zayo zangoku, i-Coluracetam ibonise amandla kunyango lweengxaki ze-neurodeergenerative ezifana nesifo se-Alzheimer kunye nokuphazamiseka kwengqondo.Uphando lucebisa ukuba i-Coluracetam inokuba neepropathi ze-neuroprotective, iyenza ibe ngumviwa onomdla wokuphononongwa ngakumbi kwezi meko.Nangona kunjalo, izifundo ezongezelelweyo kunye novavanyo lweklinikhi luyafuneka ukumisela ukusebenza kwayo, ukhuseleko, kunye neendlela ezichanekileyo zokusetyenziswa kwiisetingi zeklinikhi.

Abemi abalupheleyo banyuse imfuno yongenelelo ngoncedo olunokunciphisa ukuhla kwengqondo okunxulumene neminyaka.Imiphumo ye-neuroprotective ye-Coluracetam kunye namandla okuxhasa iindlela zokulungisa i-neural yenza kube yindlela enomdla yophando ekujonganeni nokuncipha kwengqondo okuhambelana nokuguga.

Ukongezelela, uphando lwangaphambili lubonisa ukuba i-Coluracetam ingaba neenzuzo zokuphazamiseka kwemizwelo njengokudandatheka kunye nokuxhalaba.Nangona kunjalo, uphando olubanzi ngakumbi luyafuneka ukuvavanya ukusebenza kwayo kunye nokuseka iiprothokholi zonyango ezifanelekileyo kwezi zibonakaliso.

Ikhono leColuracetam linabela kwiinkqubo ze-neurorehabilitation ngokunjalo.Ikhono layo lokuphucula ukubonakaliswa kwe-neuronal kunye nenkxaso enokuthi ixhase iindlela zokulungisa i-neural yenza ukuba ibe ngumgqatswa wokusetyenziswa ekubuyiseleni abantu abanokulimala kwengqondo okanye imivimbo.

Nangona i-Coluracetam ibonisa isithembiso kwizicelo ezahlukahlukeneyo, kubalulekile ukugxininisa imfuno yophando olongezelelweyo, ukuqinisekisa ukusebenza kwayo, ukhuseleko, kunye neendlela ezifanelekileyo zokusetyenziswa.Ulwamkelo olulawulayo luya kufuneka kusetyenziso lwayo lwezonyango kwizalathisi ezithile.


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