ibhena_yephepha

imveliso

Umenzi womgubo weColuracetam Inombolo yeCAS: 135463-81-9 Ubumsulwa obuyi-99% ubuncinci bezithako ezongezelelweyo

Inkcazo emfutshane:

I-Coluracetam lilungu losapho lwe-racetam lwee-nootropic compounds kwaye ikwaziwa ngokuba yi-MKC-231. Yaphuhliswa yiKobe Pharmaceutical Company eJapan ngenjongo yokunyanga i-AD kunye nokuphazamiseka kwengqondo.


Iinkcukacha zeMveliso

Iithegi zeMveliso

Ividiyo yeMveliso

Iiparamitha zeMveliso

Igama lemveliso

I-Coluracetam

Elinye igama

I-MKC-231;

I-2-oxo-N-(5,6,7,8-tetrahydro-2,3-dimethyl-furo[2,3-b]quinolin-4-yl)-1-pyrrolidineacetamide

Inombolo ye-CAS

135463-81-9

Ifomula yemolekyuli

C19H23N3O3

Ubunzima be-molecular

341.4

Ubunyulu

99.0%

Inkangeleko

Umgubo omhlophe

Isicelo

Isongezelelo sokutya Izinto eziluhlaza

Intshayelelo yemveliso

I-Coluracetam, ilungu losapho lwe-racemate lwee-nootropic compounds, ekwaziwa ngokuba yi-MKC-231, yi-nootropic compound eneziphumo zokukhulisa ingqondo kunye nokukhusela imithambo-luvo. I-Coluracetam isebenza ngokuguqula inkqubo ye-cholinergic. Kucingelwa ukuba inyusa amanqanaba e-acetylcholine, i-neurotransmitter ephambili kwingqondo edibene nokufunda kunye nemisebenzi yememori. I-Coluracetam yenza oku ngokunyusa inani kunye nomsebenzi we-choline uptake transporters, ngaloo ndlela iphucula ukukhululwa kwe-acetylcholine kunye nokuphucula imiqondiso phakathi kwee-neurons. Ezinye izifundo zokuqala zovavanyo kunye nezilwanyana zibonisa ukuba i-Coluracetam ineziphumo ezinokubangela ukhuseleko lwengqondo kunye nokuphucula ingqondo. Ezinye izifundo zifumanise ukuba i-Coluracetam inefuthe elithile lokuphucula ukukhubazeka kwememori kwiimodeli ze-AD.

Uphawu

(1) Ubumsulwa obuphezulu: I-Coluracetam ilungiswa kusetyenziswa iinkqubo eziphambili zokukhupha kunye nokuvelisa ukuqinisekisa ubumsulwa obuphezulu. Olu bumsulwa buphezulu lunceda ukuphucula ukufumaneka kwezinto eziphilayo kunye nokunciphisa ukwenzeka kweempembelelo ezimbi.
(2) Ukhuseleko: I-Coluracetam ithathwa njengekhuselekileyo ebantwini. Inani elikhulu lezifundo liye labonisa ukuba inetyhefu ephantsi kwaye ineziphumo ebezingalindelekanga ezincinci ngaphakathi koluhlu lwedosi olucetyiswayo.
(3) Uzinzo: Amalungiselelo eColuracetam abonisa uzinzo olugqwesileyo kwaye anokugcina umsebenzi wawo kunye nokusebenza kakuhle phantsi kweemeko ezahlukeneyo kunye neemeko zokugcina. Olu zinzo luqinisekisa ukusebenza okuzinzileyo nokuthembekileyo kwixesha elide.

Izicelo

I-Coluracetam okwangoku isetyenziswa kwiindlela ezahlukeneyo zokusebenza kwaye ibonisa ithemba elikhulu kwixesha elizayo. Isetyenziswa ngokuyintloko njengesongezelelo sokutya esiphucula ingqondo kwaye ifunwa ngabantu abafuna ukuphucula inkumbulo, ukugxila, kunye nobuchule bokufunda. Amandla ekhompawundi okuguqula inkqubo ye-cholinergic kucingelwa ukuba anegalelo kwimiphumo yayo yokuphucula ingqondo. Ukongeza, uphando lubonisa ukuba i-Coluracetam inokuba neempawu zokukhusela imithambo-luvo ezinokunceda ukuthintela ukwehla kwengqondo okunxulumene nobudala kunye nokuxhasa impilo yengqondo iyonke.


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