ibhena_yephepha

imveliso

Umenzi womgubo we-PRL-8-53 Inombolo ye-CAS: 51352-87-5 Ubumsulwa obuyi-98% ubuncinane bezithako ezongezelelweyo

Inkcazo emfutshane:

I-PRL-8-53 sisithambisi esitsha sokuqiqa, ikhompawundi ekhusela inkqubo yemithambo-luvo. Ekuqaleni yaphuhliswa nguGqr. Milton V.


Iinkcukacha zeMveliso

Iithegi zeMveliso

Iiparamitha zeMveliso

Igama lemveliso

I-PRL-8-53

Elinye igama

I-Methyl 3-(2-(benzyl(Methyl)aMino)ethyl)benzoate hydrochloride;Benzoic acid, 3-[2-[methyl(phenylmethyl)amino]ethyl]-, i-methyl ester, i-hydrochloride (1:1);I-Methyl 3-{2-[benzyl(methyl)amino]ethyl}benzoate hydrochloride (1:1)

Inombolo ye-CAS

51352-87-5

Ifomula yemolekyuli

C18H22I-ClNO2

Ubunzima be-molecular

319.83

Ubunyulu

98.0%

Inkangeleko

Umgubo omhlophe

Ukupakisha

1 kg ngebhegi nganye 25kg/idrama

Isicelo

i-nootropic

Intshayelelo yemveliso

I-PRL-8-53, eyaziwa ngokuba yi-methyl 3-(2-(benzyl(methyl)amino)ethyl)benzoate, yi-compound ye-nootropic eyenziweyo ecingelwa ukuba iphucula ukudluliselwa kwe-cholinergic kwaye ilawula amanqanaba e-dopamine engqondweni. Ezi ndlela zokuziphatha zinegalelo kwiziphumo zayo ezinokubangela ukuphuculwa kwengqondo, ngaloo ndlela ziphucula ukwakheka kwememori, ukugcinwa kwayo, kunye nokufunyanwa kwayo. Izifundo ezininzi kwizilwanyana nakubantu zibike iziphumo ezilungileyo zeempawu zayo zokuphucula imemori. Kwisifundo sovavanyo olulawulwa yi-placebo, abantu abafumene idosi enye ye-PRL-8-53 babonise inkumbulo yamagama engcono kunye nokukwazi ukufumana ulwazi xa kuthelekiswa neqela le-placebo. Ezi ziphumo zivuse umdla kunye nophando olongezelelekileyo malunga nokukwazi kwe-compound. Olunye uphando kwiimpuku lubonise ukuba ukunika i-PRL-8-53 kuphucule kakhulu amandla azo okufunda kumsebenzi we-maze wamanzi. Iimpuku eziphathwe nge-PRL-8-53 zikwazile ukufumana iqonga elifihliweyo ngokufanelekileyo kunezolawulo, zibonisa amandla e-compound njengokuphucula imemori.

Uphawu

(1) Ubunyulu obuphezulu: I-PRL-8-53 inokufumana iimveliso ezinyulu obuphezulu ngokusebenzisa iinkqubo zemveliso zokucoca. Ubunyulu obuphezulu buthetha ukufumaneka ngcono kwezinto eziphilayo kunye neempendulo ezimbalwa ezingalunganga.

(2) Ukhuseleko: Ukhuseleko oluphezulu, zimbalwa iziphumo ezimbi, akukho ziphumo ezimbi zicacileyo.

(3) Uzinzo: I-PRL-8-53 izinzile kakuhle kwaye inokugcina umsebenzi wayo kunye nesiphumo phantsi kweemeko ezahlukeneyo kunye neemeko zokugcina.

Izicelo

Njengohlobo olutsha lwesongezelelo sokuphucula ingqondo, i-PRL-8-53 iphucula inkumbulo yexesha elifutshane kunye nenkumbulo yokusebenza, ngelixa iphucula amandla okufunda kunye nesantya sokufumana izakhono, inceda ekuphuculeni ukufunda kunye nokusebenza kakuhle. Uphando lubonisa ukuba i-PRL-8-53 inokukhuthaza ukukhula kunye nokuvuselelwa kwee-neurons engqondweni. I-PRL-8-53 inokunyusa isantya apho ingqondo icubungula ulwazi, ivumela abantu ukuba bagqibe imisebenzi kwaye benze izigqibo ngokukhawuleza. Nangona ithelekiswa nezinye iikhompawundi ze-nootropic Nangona kunjalo, uphando kwi-PRL-8-53 lulinganiselwe, kodwa uphando olukhoyo lubonisa amandla ayo okuphucula inkumbulo kunye nezakhono zokuqonda.


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