I-Compound 7P umenzi we powder CAS No.: 1890208-58-8 99% ubumsulwa min.zokongeza izithako
IiParameters zeMveliso
Igama lemveliso | I-Compound 7P |
Elinye igama | Compound7P;2- [(2-methoxyphenyl)[(4-methylphenyl)sulfonyl]amino]-N-(4-methoxy-3-pyridinyl)acetamide; 2-(N-(2-methoxyphenyl) -4-methylphenylsulfonamido)-N-(4-methoxypyridin-3-yl)acetamide |
Inombolo yeCAS. | 1890208-58-8 |
Ifomula yemolekyuli | I-C22H23N3O5S |
Ubunzima bemolekyuli | 441.51 |
Ubunyulu | 99.0% |
Imbonakalo | Umgubo omhlophe |
Isicelo | Nootropic |
Intshayelelo yemveliso
I-Compound 7p iboniswe ukukhuthaza ukukhula kwe-GAP-43-positive axons kwimodeli yezilwanyana zokulimala kwe-nerve optic, ebonisa ukuba umsebenzi we-neurite outgrowth we-compound 7p in vitro uguqulela ekukhuthazeni ukuvuselelwa kwe-axon kwi-vivo.I-Compound 7P powder iyimpuphu emhlophe emhlophe eveliswa njenge-tandem compound yokuchonga i-dual-acting thromboxane receptor antagonist inhibitors.Enyanisweni, i-compound 7p ibonisa ukukhetha kwe-prostaglandin I2 synthase (PTGIS, CYP8A1) phezu kwe-thromboxane synthase (CYP5A1).I-nootropic yiyo nayiphi na into enceda ukuphucula ukusebenza kwengqondo, kuquka imemori, ukugxininiswa, isimo sengqondo, kunye nobukrelekrele.Zinokusuka kumaqela athile okutya okanye izinto ukuya kwiikhompawundi ezenziwe ngabantu ezilungiselelwe ngokukodwa ukunceda ukusebenza kwengqondo kunye nezinye izibonelelo.I-Nootropic compound 7P powder ikhuthaza ukuphuma kwe-Gap-43 i-axons emihle, ngaloo ndlela ivuselela ukuvuselelwa kwe-axonal kwi-vivo.I-7p yekhwalithi ephezulu yenzelwe ukuphucula ukulungelelaniswa, ukuphucula isimo sengqondo kunye nokunceda ukulwa nokudinwa.Ikwanqanda i-oxidation yengqondo kwaye inceda ukulwa nomonakalo wobuchopho obangelwa kukusetyenziswa kotywala.
Usetyenziso
I-Neurons kwinkqubo ye-nervous central (CNS) iyasilela ukuhlaziya i-axon emva kokulimala, okuyingxenye echaza ukubuyiswa kokusebenza kakubi kwizigulane ezine-trauma kunye nezifo ze-neurodeergenerative.I-Compound 7p, ephucula ukuphuma kwe-neurite kwii-neurons eziphambili ezikhuliswe kwi-hippocampus, i-cortex ye-cerebral, kunye ne-retina, kwaye ibangele ukuvuselelwa kwe-nerve ye-optic kwimodeli yezilwanyana yokulimala kwe-optic nerve.Ikwanyusa ulungelelwaniso, iphatha ukonakala kwengqondo okunxulumene notywala, kwaye inqande i-oxidation ejikeleze ingqondo.Kwakhona kunceda ukuphucula isimo sengqondo kunye nokulwa nokudinwa.Ukongeza i-7P edibeneyo ibonise owona msebenzi uphezulu ngokuchasene namathumba omlomo wesibeleko ngokuphucula i-microstructure ngendlela exhomekeke kwidosi.Ukulungiswa ngakumbi kwe-compound 7p kunye nokucaciswa kwendlela ebangela ngayo ukuvuselelwa kwe-axon kwi-vivo kuya kubonelela ngengqiqo kwiinzame zexesha elizayo zokuqinisa izicwangciso zonyango.