Umenzi womgubo weCompound 7P Inombolo yeCAS: 1890208-58-8 Ubumsulwa obuyi-99% ubuncinane bezithako ezongezelelweyo
Ividiyo yeMveliso
Iiparamitha zeMveliso
| Igama lemveliso | I-Compound 7P |
| Elinye igama | I-Compound7P;2-[(2-methoxyphenyl)[(4-methylphenyl)sulfonyl]amino]-N-(4-methoxy-3-pyridinyl)acetamide; 2-(N-(2-methoxyphenyl)-4-methylphenylsulfonamido)-N-(4-methoxypyridin-3-yl)acetamide |
| Inombolo ye-CAS | 1890208-58-8 |
| Ifomula yemolekyuli | C22H23N3O5S |
| Ubunzima be-molecular | 441.51 |
| Ubunyulu | 99.0% |
| Inkangeleko | Umgubo omhlophe |
| Isicelo | I-Nootropic |
Intshayelelo yemveliso
I-Compound 7P ibhekisa kwi-organic compound ethile equlethe ii-athomu zekhabhoni ezisixhenxe. Kwi-organic chemistry, ikhabhoni yinto ebalulekileyo kuba inokwenza amakhonkco azinzileyo nezinye ii-athomu, kuquka ii-athomu zekhabhoni, ukuze zenze ii-molecules ezintsonkothileyo. Ezi molekyuli zinokuba neepropati ezahlukeneyo kunye nemisebenzi, zenze ii-compounds ezisekelwe kwikhabhoni zibe zizinto zokwakha ubomi. Kwiimodeli zezilwanyana zokwenzakala kwe-optic nerve, i-compound 7p iboniswe ukuba ikhuthaza ukukhula kwee-axons ze-GAP-43-positive, nto leyo ebonisa ukuba umsebenzi wokukhula kwe-neurite we-compound 7p in vitro uguqulela ekukhuthazeni ukuvuselelwa kwe-axonal in vivo. I-Compound 7P powder yi-white to off-white powder eveliswa njenge-tandem compound yokuchonga ii-antagonist inhibitors ze-thromboxane receptor antagonist. Enyanisweni, i-compound 7p ibonise ukukhetha kwe-prostaglandin I2 synthase (PTGIS, CYP8A1) xa kuthelekiswa ne-thromboxane synthase (CYP5A1). I-nootropic compound 7P powder ikhuthaza ukukhula kwee-axons ze-Gap-43-positive, ngaloo ndlela ivuselela ukuvuselelwa kwe-axonal emzimbeni. I-Complex 7p esemgangathweni ophezulu yenzelwe ukuphucula ulungelelwaniso, ukuphucula imeko yeemvakalelo kunye nokunceda ukulwa nokudinwa. Ikwathintela ukubola kwengqondo kwaye inceda ukulwa nomonakalo wengqondo obangelwa kukusela utywala.
Uphawu
(1) Ubunyulu obuphezulu: I-Compound 7P inokufumana iimveliso ezinyulu obuphezulu ngeenkqubo zemveliso ezicociweyo. Ubunyulu obuphezulu buthetha ukufumaneka ngcono kwezinto eziphilayo kunye neempendulo ezimbalwa ezingalunganga.
(2) Ukhuseleko: I-Compound 7P ibonakalisiwe ukuba ikhuselekile emzimbeni womntu.
(3) Uzinzo: I-Compound 7P inozinzo oluhle kwaye ingagcina umsebenzi wayo kunye nesiphumo phantsi kweemeko ezahlukeneyo kunye neemeko zokugcina.
Izicelo
I-Compound 7p iphucula ukukhula kwe-neurite kwii-neurons eziphambili ezikhuliswe kwi-hippocampus, i-cerebral cortex, kunye ne-retina kwaye ikhuthaza ukuvuselelwa kwe-optic nerve kwiimodeli zezilwanyana zokwenzakala kwe-optic nerve. Ikwaphucula ukulungelelaniswa, inyanga umonakalo wengqondo onxulumene notywala, kwaye ithintele i-oxidation ejikeleze ingqondo. Ikwanceda ukuphucula imo yengqondo kunye nokulwa nokudinwa.












