I-Amino Tadalafil powder umenzi we-CAS No.: 385769-84-6 98% ubumsulwa min. zokongeza izithako
Ividiyo yeMveliso
Iiparamitha zeMveliso
Igama lemveliso | Amino Tadalafil |
Elinye igama | (6R,12aR)-2-Amino-6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[ 3,4-b]indole-1,4-dione;AminoTadalafil(6R,12Ar)-2-Amino-6-(1,3-Benzodioxol-5-Yl)-2,3,6,7,12,12A -Hexahydropyrazino [1',2':1,6]Pyrido[3,4-B]Indole-1,4-Dione;(6R,12aR) -2-Amino-6-(benzo[d][1,3] ]dioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indol-1,4-dione;(6R ,12aR) -2-amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,12,12a-tetrahydropyrazino[1',2':1,6]pyrido[3] ,4-b]indole-1,4(6H,7H)-dione |
Inombolo yeCAS. | 385769-84-6 |
Ifomula yemolekyuli | I-C21H18N4O4 |
Ubunzima bemolekyuli | 390.39 |
Ubunyulu | 98.0% |
Imbonakalo | Umgubo omhlophe ukuya kumhlophe |
Isicelo | I-Dietary Supplement Raw Material |
Intshayelelo yemveliso
I-Amino Tadalafil yikhompawundi entsha, i-derivative ye-tadalafil, eya isanda kakhulu kwintsimi ye-erectile dysfunction (ED). Idibanisa i-amino acid kunye ne-tadalafil, i-FDA-evunyiweyo ye-PDE5 inhibitor eyona nto isetyenziselwa ukuphatha i-ED. Isebenza ngokunyusa ukuhamba kwegazi kwi-penis, ukuvumela amadoda ukuba afezekise kwaye agcine i-erection. Ii-amino acids, kwelinye icala, zidlala indima ebalulekileyo kwimisebenzi eyahlukeneyo yomzimba, kubandakanywa ukuveliswa kweeprotheni, ezizibhloko zokwakha izicubu kunye namalungu. Ukudibanisa kwezi zimbini izithako zenzelwe ukuphucula ukusebenza kweTadalafil ekuphatheni i-ED. Kwaye i-amino Tadalafil yinguqulo ephuculweyo enamandla angaqhelekanga, ephucula ukusebenza kunye nokuguquguquka kwangaphambi kwayo. Ubume bayo beekhemikhali buhlala bufana neTadalafil, kodwa ngokusungulwa kwamaqela e-amino, ifumana iimpawu ezikhethekileyo ezenza ukuba zivelele kwihlabathi lamachiza. Njenge-tadalafil, i-Amino Tadalafil isebenza ngokuvimbela i-phosphodiesterase 5 (PDE5), i-enzyme ejongene nokuphula i-cyclic guanosine monophosphate (cGMP) emzimbeni. I-cGMP yikhompawundi yendalo ekhuthaza ukukhululeka kwemithambo yegazi, ngaloo ndlela inyusa ukuhamba kwegazi. Ngokuthintela i-PDE5, i-amino Tadalafil iqinisekisa ukuqokelela kwe-cGMP, ngaloo ndlela iphucula i-vasodilation kunye nokuphucula ukujikeleza kwegazi. Ukongezelela, abaphandi baye bahlola amandla ayo okunceda ukunyanga i-benign prostatic hyperplasia (BPH) ngokukhuthaza ukuhamba kwegazi kwi-prostate.
Uphawu
(1) Ukucoceka okuphezulu: I-Amino Tadalafil inokufumana iimveliso ezicocekileyo ngokucokisa iinkqubo zokuvelisa. Ukucoceka okuphezulu kuthetha ukuba ngcono kwe-bioavailability kunye neempendulo ezimbalwa ezimbi.
(2) Ukhuseleko: Ukhuseleko oluphezulu, iimpendulo ezimbalwa ezimbi.
(3) Ukuzinza: I-Amino Tadalafil inozinzo oluhle kwaye inokugcina umsebenzi wayo kunye nesiphumo phantsi kweemeko ezahlukeneyo kunye neemeko zokugcina.
Usetyenziso
I-Amino Tadalafil yi-PDE5 inhibitor enemiphumo efanayo ye-pharmacological njenge-tadalafil. Ngokudibanisa i-amino acids kunye ne-tadalafil, i-amino Tadalafil icingelwa ukuba isebenze ngakumbi ekuphatheni i-erectile dysfunction kune-tadalafil yodwa. Ii-amino acids zinokunceda ukunyusa ukujikeleza kwegazi kunye nokuxhasa ukusebenza ngokupheleleyo kwamayeza. Ukongezelela, inokuphucula iimpawu ze-erectile dysfunction (ED) ngokuthintela umsebenzi we-PDE5 enzyme ukukhuthaza ukuhamba kwegazi kwizitho zokuzala zesilisa. Xa kuthelekiswa ne-tadalafil, i-amino Tadalafil i-metabolized ngokuthe ngcembe emzimbeni kwaye inokuvelisa iziphumo ezihlala ixesha elide. Oku kunika i-amino Tadalafil amandla amakhulu ekuphatheni i-ED.