Umenzi womgubo we-OTR-AC(Ostarine Acetate) 98% ubumsulwa bomda kwizithako ezongezelelweyo
Iiparamitha zeMveliso
| Igama lemveliso | I-OTR-AC |
| Elinye igama | I-Ostarine Acetate |
| Ifomula yemolekyuli | C21H16F3N3O4 |
| Ubunzima be-molecular | 431.36 |
| Ubunyulu | 98.0% |
| Inkangeleko | Umgubo omhlophe |
| Ukupakisha | 1kg/ibhegi 25kg/igubu |
| Isicelo | Fumana izihlunu kwaye unciphise amafutha |
Intshayelelo yemveliso
I-OTR-AC, eyaziwa ngokuba yi-MK-2866 Ester, yi-MK-2866 (i-Ostarine) eye yafumana i-esterification (inkqubo yokudibanisa i-organic acid kunye ne-alcohol). Le nkqubo yekhemikhali isetyenziselwa ukwandisa amandla esinto kunye nokwandisa isiqingatha sobomi (ixesha elithathayo ukuba isixa sehle siye kwisiqingatha sexabiso laso lokuqala). Ngenxa yale nkqubo, inguqulelo ye-ester ye-ostarine inamandla aphindwe kalishumi okugcina umsebenzi webhayoloji. Oku kufezekisa iingenelo ezongezelelweyo, njengenguqulelo ye-ester ye-selective androgen receptor modulator (SARM) Ostarin, i-OTR-AC inamandla ngakumbi kwaye ihlala ixesha elide. Ngokunamathela kwiproteni emzimbeni ebizwa ngokuba yi-androgen receptor, ivuselela ukwakheka kwezicubu zemisipha. Oku kwandisa ubunzima bemisipha kunye namandla.
Uphawu
(1) Ubunyulu obuphezulu: I-OTR-AC inokufumana iimveliso ezinyulu obuphezulu ngeenkqubo zokuvelisa ezicociweyo. Ubunyulu obuphezulu buthetha ukufumaneka ngcono kwezinto eziphilayo kunye neempendulo ezimbalwa ezingalunganga.
(2) Ukhuseleko: I-OTR-AC yimveliso yendalo ebonakaliswe ikhuselekile emzimbeni womntu.
(3) Uzinzo: I-OTR-AC izinzile kakuhle kwaye inokugcina umsebenzi wayo kunye nesiphumo phantsi kweemeko ezahlukeneyo kunye neemeko zokugcina.
Izicelo
I-OTR-AC isebenza njenge-selective androgen receptor modulator (SARM), oko kuthetha ukuba isebenza ngokukhetha kwizicubu zemisipha kunye nezicubu zamathambo emzimbeni ngaphandle kokuchaphazela amanye amalungu kunye nezicubu. Iphucula ubunzima bemisipha kunye nokusebenza komzimba, inceda ukwandisa ubunzima bemisipha kunye namandla ngelixa inciphisa umxholo wamafutha. I-OTR-AC isebenza nezinye ii-SARM ukwandisa ubunzima bemisipha kunye namandla ngokuvuselela ukwakheka kwezicubu zemisipha. Ukongeza ekuncedeni ukwandisa ubunzima bemisipha, i-OTR-AC ifunyenwe inciphisa amafutha omzimba ngokubanzi. I-OTR-AC iyanda ngokuphucula imetabolism ye-lipid kunye nokuchaphazela ukukhululwa kwe-adiponectin, i-hormone elawula ukuqhekeka kwamafutha acids Ukuqhekeza iiseli zamafutha, i-OTR-AC inokunceda ekuvuseleleni ukwakheka kwamathambo kunye nokuthintela izifo zamathambo.












